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Mutant IDH1 inhibitor
CAS No. 1429180-08-4
Mutant IDH1 inhibitor( —— )
Catalog No. M23590 CAS No. 1429180-08-4
Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 151 | In Stock |
|
| 10MG | 259 | In Stock |
|
| 25MG | 437 | In Stock |
|
| 50MG | 624 | In Stock |
|
| 100MG | 888 | In Stock |
|
| 500MG | 1773 | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameMutant IDH1 inhibitor
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NoteResearch use only, not for human use.
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Brief DescriptionMutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
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DescriptionMutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
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In VitroMutant IDH1 inhibitor is a potent IDH1 R132H inhibitor, and used for the treatment of diseases or disorders associated with such mutant IDH proteins including, but not limited to, cell-proliferation disorders, such as cancer.
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In Vivo——
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Synonyms——
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PathwayMetabolic Enzyme/Protease
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TargetDehydrogenase
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Recptormutant IDH1 R132H
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Research Area——
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Indication——
Chemical Information
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CAS Number1429180-08-4
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Formula Weight466.58
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Molecular FormulaC25H34N6O3
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Purity>98% (HPLC)
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SolubilityDMSO:30 mg/mL (64.3 mM)
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SMILESCC(C)[C@@H](COC1=O)N1c1nc(N[C@@H](C)c2ccc(CN(CC3)CCN3C(C)=O)cc2)ncc1
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.3-Pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH and their preparation. Patent WO 2013046136 A1 20130404
molnova catalog
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