Mutant IDH1 inhibitor

CAS No. 1429180-08-4

Mutant IDH1 inhibitor( —— )

Catalog No. M23590 CAS No. 1429180-08-4

Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 151 In Stock
10MG 259 In Stock
25MG 437 In Stock
50MG 624 In Stock
100MG 888 In Stock
500MG 1773 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    Mutant IDH1 inhibitor
  • Note
    Research use only, not for human use.
  • Brief Description
    Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
  • Description
    Mutant IDH1 inhibitor is an effective inhibitor of mutant IDH1 R132H (IC50: < 72 nM).
  • Synonyms
    ——
  • Pathway
    Metabolic Enzyme/Protease
  • Target
    Dehydrogenase
  • Recptor
    mutant IDH1 R132H
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1429180-08-4
  • Formula Weight
    466.6
  • Molecular Formula
    C25H34N6O3
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:30 mg/mL (64.3 mM)
  • SMILES
    CC(C)[C@@H](COC1=O)N1c1nc(N[C@@H](C)c2ccc(CN(CC3)CCN3C(C)=O)cc2)ncc1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.3-Pyrimidin-4-yl-oxazolidin-2-ones as inhibitors of mutant IDH and their preparation. Patent WO 2013046136 A1 20130404
molnova catalog
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